Inhibidores de entrada vih (yo)
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INHIBIDORES DE ENTRADA • Inhibidores de unión • Inhibidores de correceptores • Inhibidores de fusión DARYA HUANCHACO NUÑEZ.
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Transcript of Inhibidores de entrada vih (yo)
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INHIBIDORES DE ENTRADA• Inhibidores de unión
• Inhibidores de correceptores
• Inhibidores de fusión
DARYA HUANCHACO NUÑEZ.
![Page 2: Inhibidores de entrada vih (yo)](https://reader036.fdocuments.ec/reader036/viewer/2022081519/55b18752bb61ebb44a8b456e/html5/thumbnails/2.jpg)
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Inhibidores de unión
![Page 5: Inhibidores de entrada vih (yo)](https://reader036.fdocuments.ec/reader036/viewer/2022081519/55b18752bb61ebb44a8b456e/html5/thumbnails/5.jpg)
Inhibidores de correceptores: CXCR4 y CCR5
Inhibidores de entrada: Maravicoc ( Selzentry)
![Page 6: Inhibidores de entrada vih (yo)](https://reader036.fdocuments.ec/reader036/viewer/2022081519/55b18752bb61ebb44a8b456e/html5/thumbnails/6.jpg)
Inhibidores de fusión: Enfuvirtide( Fuzeon) Detiene el VIH en e punto de fusión, antes de que acceda a la célula
GP41
• La gp41 consta de 3 dominios• El ectodominio tiene 3 unidades
funcionales• Regiones hidrofóbicas, HR1 y HR2.• La gp 41 zipping “cierre de cremalleras”• Enfuvirtide imita la región HR2 de la
gp41
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¡GRACIAS!